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Nicardipine: Mechanism, Uses, and Administration

Writer's picture: MaytaMayta

Updated: Jan 28

Nicardipine IV Drip Protocol Concentration

  • Mix 20 mg of nicardipine in 80 mL to 100 mL of normal saline (NSS).

  • This results in a concentration of 0.2 mg/mL.

Infusion Rate

  • Administer between 10-70 mL/hour, adjusting based on the patient's blood pressure and clinical condition.

  • Titrate by 5 mL/hour every 5-15 minutes to achieve the desired systolic blood pressure (SBP).


Target SBP

  • Maintain systolic blood pressure (SBP) ≤ 160 mmHg (adjust further based on specific clinical scenarios or comorbidities).

  • In hypertensive emergencies, aim to reduce mean arterial pressure (MAP) by no more than 25% within the first hour, then a gradual reduction over the next 2-6 hours.


 

Mechanism of Action

Nicardipine is a dihydropyridine calcium channel blocker that acts as a vasodilator to lower blood pressure by:

  1. Blocking L-type calcium channels: Inhibits calcium influx, primarily in vascular smooth muscle cells.

  2. Inducing arterial vasodilation: Reduces systemic vascular resistance (afterload), effectively decreasing blood pressure.


 

Indications

Nicardipine is primarily indicated for:

  • Hypertensive emergencies

  • Chronic hypertension (oral formulation)

  • Angina pectoris: Dilates coronary arteries, improving myocardial oxygen supply.


 

Comparison with Other Calcium Channel Blockers

  • Verapamil/Diltiazem: Affect cardiac conduction and heart rate, making them suitable for atrial fibrillation or arrhythmia management.

  • Nicardipine: Lacks significant action on the sinoatrial (SA) or atrioventricular (AV) nodes, focusing instead on vascular effects.


 

Preparation and Administration

  1. Preparation

    • Mix 20 mg of nicardipine in 80-100 mL NSS (0.2 mg/mL).

    • Ensure thorough mixing of the solution.

  2. Administration

    • Start infusion at 10-15 mL/hour.

    • Titrate by 5 mL/hour every 5-15 minutes to achieve the target BP.

    • Maximum rate: 70 mL/hour.

Example Dose Calculation

  • Initial Rate: 15 mL/hour = 3 mg/hour.

  • Adjustment: Increase to 20 mL/hour = 4 mg/hour.

  • Max Dose: 70 mL/hour = 14 mg/hour.


 

Monitoring and Safety

  1. Blood Pressure and Heart Rate

    • Continuous monitoring is critical.

    • Avoid overshooting target BP, which can result in hypotension.

  2. Infusion Site

    • Monitor for signs of phlebitis or extravasation.


 

Common Side Effects

  • Hypotension: Excessive vasodilation.

  • Reflex tachycardia: Compensatory mechanism for decreased BP.

  • Headache, flushing, dizziness: Due to systemic vasodilation.


 

Key Considerations

  • Use an IV pump for precise control of infusion rates.

  • Individualize BP targets based on patient-specific factors.

  • Gradual adjustment is essential to prevent ischemia or other complications.

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